Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,111
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1,111
Tocris Bioscience™ CyPPA
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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KCa2.2 and KCa2.3 (SK) channel activator
| CAS | 73029-73-9 |
|---|---|
| Chemical Name or Material | N-Cyclohexyl-N-[2-(3,5-dimethyl-pyrazol-1-yl)-6-methyl-4-pyrimidinamine |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C16H23N5 |
| Formula Weight | Observed MW: 285.39 |
| Assay Percent Range | >99% |
1,112
Tocris Bioscience™ cAMPS-Rp, triethylammonium salt
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CAS: 151837-09-1 Molecular Formula: C16H27N6O5PS
| CAS | 151837-09-1 |
|---|---|
| Molecular Formula | C16H27N6O5PS |
1,113
| Target | Muscarinic Acetylcholine Receptor M5/CHRM5 |
|---|---|
| CAS | 2926782-31-0 |
| Purity | 0.98 |
| Chemical Name or Material | (3R,4S)-rel-1-[(2,3-Dihydro-5-benzofuranyl)sulfonyl]-3-fluoro-4-[[(1-methyl-1H-imidazol-2-yl)thio]methyl]piperidine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H22FN3O3S2 |
1,114
Tocris Bioscience™ YE 120
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 383124-82-1 Molecular Formula: C16H9Cl2N3O
| CAS | 383124-82-1 |
|---|---|
| Molecular Formula | C16H9Cl2N3O |
1,115
Tocris Bioscience™ PD 168077 maleate
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CAS: 630117-19-0 Molecular Formula: C24H26N4O5
| CAS | 630117-19-0 |
|---|---|
| Molecular Formula | C24H26N4O5 |
1,116
| Target | Adrenergic alpha-2 Receptor Antagonists |
|---|---|
| CAS | 2313483-41-7 |
| Purity | 0.98 |
| Chemical Name or Material | 1-[2-[[[3-(3,5-Dimethyl-4-isoxazolyl)imidazo[1,2-a]pyridin-7-yl]carbonyl]amino]ethyl]-4-(methylamino)pyridinium chloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H23ClN6O2 |
1,117
Tocris Bioscience™ Dihydrokainic acid
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CAS: 52497-36-6 Molecular Formula: C10H17NO4
| CAS | 52497-36-6 |
|---|---|
| Molecular Formula | C10H17NO4 |
1,118
Tocris Bioscience™ SRT 1720
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Selective SIRT1 activator; induces autophagy and mitochondrial biogenesis
| Target | Sirtuin 1/SIRT1 |
|---|---|
| CAS | 925434-55-5 |
| Purity | 0.98 |
| Chemical Name or Material | N-[2-[3-(1-Piperazinylmethyl)imidazo[2,1-b]thiazol-6-yl]phenyl]-2-quinoxalinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H23N7OS |
1,119
Tocris Bioscience™ TFC 007
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Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
| Inhibitors | TFC 007 |
|---|---|
| Product Type | TFC 007 |
| Molecular Weight (g/mol) | 487.55 |
| Purity | >98% |
1,120
Tocris Bioscience™ LY 354740
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 176199-48-7 Molecular Formula: C8H11NO4
| CAS | 176199-48-7 |
|---|---|
| Molecular Formula | C8H11NO4 |
1,121
Tocris Bioscience™ BPTU
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P2Y1 allosteric antagonist
| CAS | 870544-59-5 |
|---|---|
| Chemical Name or Material | N-[2-[2-(1,1-Dimethylethyl)phenoxy]-3-pyridinyl]-N′-[4-(trifluoromethoxy)phenyl]urea |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C23H22F3N3O3 |
| Formula Weight | Observed MW: 445.43 |
| Assay Percent Range | >98% |
1,122
Tocris Bioscience™ Mpro Tracer
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SARS-CoV-2 main protease fluorescent ligand; TR-FRET acceptor
1,123
Tocris Bioscience™ L-371,257
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CAS: 162042-44-6 Molecular Formula: C28H33N3O6
| CAS | 162042-44-6 |
|---|---|
| Molecular Formula | C28H33N3O6 |
1,124
Tocris Bioscience™ Clozapine
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CAS: 5786-21-0 Molecular Formula: C18H19ClN4
| CAS | 5786-21-0 |
|---|---|
| Molecular Formula | C18H19ClN4 |
1,125
Tocris Bioscience™ TRPC6-PAM-C20
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Selective TRPC6 positive allosteric modulator
| CAS | 667427-75-0 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3-(3-,4-Dihydro-6,7-dimethoxy-3,3-dimethyl-1-isoquinolinyl)-2H-1-benzopyran-2-one |
| Molecular Formula | C22H21NO4 |